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| Issue Date | Title | Author(s) |
| 2018 | 1,3,5-triazaspiro[5.5]undeca-2,4-dienes as selective Mycobacterium tuberculosis dihydrofolate reductase inhibitors with potent whole cell activity | Yang, Xuan; Wedajo, Wassihun; Yamada, Yoshiyuki; Dahlroth, Sue-Li; Neo, Jason Jun-Long; Dick, Thomas; Chui, Wai-Keung |
| 2022 | Anti-Mycobacterium abscessus activity of tuberculosis F-ATP synthase inhibitor GaMF1 | Ragunathan, Priya; Dick, Thomas; Grüber, Gerhard |
| 2020 | Antituberculosis activity of the antimalaria cytochrome bcc oxidase inhibitor SCR0911 | Chong, Sherilyn Shi Min; Manimekalai, Malathy Sony Subramanian; Sarathy, Jickky Palmae; Williams, Zoe C.; Harold, Liam K.; Cook, Gregory M.; Dick, Thomas; Pethe, Kevin; Bates, Roderick Wayland; Grüber, Gerhard |
| 2022 | Atomic solution structure of Mycobacterium abscessus F-ATP synthase subunit ε and identification of Ep1MabF1 as a targeted inhibitor | Shin, Joon; Harikishore, Amaravadhi; Wong, Chui Fann; Ragunathan, Priya; Dick, Thomas; Grüber, Gerhard |
| 2016 | Bedaquiline Targets the ε Subunit of Mycobacterial F-ATP Synthase | Kundu, Subhashri; Biukovic, Goran; Grüber, Gerhard; Dick, Thomas |
| 2016 | Deletion of a unique loop in the mycobacterial F-ATP synthase γ subunit sheds light on its inhibitory role in ATP hydrolysis-driven H+ pumping | Hotra, Adam; Suter, Manuel; Biuković, Goran; Priya, Ragunathan; Kundu, Subhashri; Dick, Thomas; Grüber, Gerhard |
| 2020 | Discovery of a novel mycobacterial F-ATP synthase inhibitor and its potency in combination with diarylquinolines | Hotra, Adam; Ragunathan, Priya; Ng, Pearly Shuyi; Seankongsuk, Pattarakiat; Harikishore, Amaravadhi; Sarathy, Jickky Palmae; Saw, Wuan-Geok; Lakshmanan, Umayal; Sae-Lao, Patcharaporn; Kalia, Nitin Pal; Shin, Joon; Kalyanasundaram, Revathy; Anbarasu, Sivaraj; Parthasarathy, Krupakar; Pradeep, Chaudhari Namrata; Makhija, Harshyaa; Dröge, Peter; Poulsen, Anders; Tan, Jocelyn Hui Ling; Pethe, Kevin; Dick, Thomas; Bates, Roderick Wayland; Grüber, Gerhard |
| 2019 | Disrupting coupling within mycobacterial F-ATP synthases subunit ε causes dysregulated energy production and cell wall biosynthesis | Saw, Wuan-Geok; Wu, Mu-Lu; Ragunathan, Priya; Biuković, Goran; Lau, Aik-Meng; Shin, Joon; Harikishore, Amaravadhi; Cheung, Chen-Yi; Hards, Kiel; Sarathy, Jickky Palmae; Bates, Roderick Wayland; Cook, Gregory M.; Dick, Thomas; Grüber, Gerhard |
| 2023 | GaMF1.39’s antibiotic efficacy and its enhanced antitubercular activity in combination with Clofazimine, Telacebec, ND-011992 or TBAJ-876 | Ragunathan, Priya; Ng, Pearly Shuyi; Singh, Samsher; Poh, Wee Han; Litty, Dennis; Kalia, Nitin Pal; Larsson, Simon; Harikishore, Amaravadhi; Rice, Scott A.; Ingham, Philip William; Müller, Volker; Moraski, Garrett; Miller, Marvin J.; Dick, Thomas; Pethe, Kevin; Grüber, Gerhard |
| 2022 | Mutational analysis of mycobacterial F‑ATP synthase subunit δ leads to a potent δ enzyme inhibitor | Harikishore, Amaravadhi; Saw, Wuan-Geok; Ragunathan, Priya; Litty, Dennnis; Dick, Thomas; Müller, Volker; Grüber, Gerhard |
| 2021 | Mycobacterium tuberculosis PanD structure-function analysis and identification of a potent pyrazinoic acid-derived enzyme inhibitor | Ragunathan, Priya; Cole, Malcolm; Latka, Chitra; Aragaw, Wassihun Wedajo; Hegde, Pooja; Shin, Joon; Manimekalai, Malathy Sony Subramanian; Rishikesan, Sankaranarayanan; Aldrich, Courtney C.; Dick, Thomas; Grüber, Gerhard |
| 2018 | The NMR solution structure of Mycobacterium tuberculosis F-ATP synthase subunit ε provides new insight into energy coupling inside the rotary engine | Joon, Shin; Ragunathan, Priya; Sundararaman, Lavanya; Nartey, Wilson; Kundu, Subhashri; Manimekalai, Malathy Sony Subramanian; Bogdanović, Nebojša; Dick, Thomas; Grüber, Gerhard |
| 2018 | Novel acetamide indirectly targets mycobacterial transporter MmpL3 by proton motive force disruption | Shetty, Annanya; Xu, Zhujun; Lakshmanan, Umayal; Hill, Jeffrey; Choong, Meng Ling; Chng, Shu-Sin; Yamada, Yoshiyuki; Poulsen, Anders; Dick, Thomas; Gengenbacher, Martin |
| 2019 | Overexpression, purification, enzymatic and microscopic characterization of recombinant mycobacterial F-ATP synthase | Saw, Wuan-Geok; Wong, Chui-Fann; Dick, Thomas; Grüber, Gerhard |
| 2020 | Pyrazinamide triggers degradation of its target aspartate decarboxylase | Gopal, Pooja; Sarathy, Jickky Palmae; Yee, Michelle; Ragunathan, Priya; Shin, Joon; Bhushan, Shashi; Zhu, Junhao; Akopian, Tatos; Kandror, Olga; Lim, Teck Kwang; Gengenbacher, Martin; Lin, Qingsong; Rubin, Eric J.; Grüber, Gerhard; Dick, Thomas |
| 2019 | Re-understanding the mechanisms of action of the anti-mycobacterial drug bedaquiline | Sarathy, Jickky Palmae; Gruber, Gerhard; Dick, Thomas |
| 2022 | Structural and mechanistic insights into Mycobacterium abscessus as-partate decarboxylase PanD and a pyrazinoic acid-derived inhibitor | Saw, Wuan Geok; Leow, Chen Yen; Harikishore, Amaravadhi; Shin, Joon; Cole, Malcolm S.; Aragaw, Wassihun Wedajo; Ragunathan, Priya; Hegde, Pooja; Aldrich, Courtney C.; Dick, Thomas; Grüber, Gerhard |
| 2022 | Structural elements involved in ATP hydrolysis inhibition and ATP synthesis of tuberculosis and non-tuberculous mycobacterial F-ATP synthase decipher new targets for inhibitors | Wong, Chui Fann; Saw, Wuan Geok; Basak, Sandip; Sano, Mio; Ueno, Hiroshi; Kerk, Hwee Wen; Litty, Dennis; Ragunathan, Priya; Dick, Thomas; Müller, Volker; Noji, Hiroyuki; Grüber, Gerhard |
| 2022 | Structure activity relationship of pyrazinoic acid analogs as potential antimycobacterial agents | Hegde, Pooja V.; Aragaw, Wassihun W.; Cole, Malcolm S.; Jachak, Gorakhnath; Ragunathan, Priya; Sharma, Sachin; Harikishore, Amaravadhi; Grüber, Gerhard; Dick, Thomas; Aldrich, Courtney C. |
| 2018 | Structure and function of Mycobacterium-specific components of F-ATP synthase subunits α and ε | Bogdanović, Nebojša; Sundararaman, Lavanya; Kamariah, Neelagandan; Tyagi, Anu; Bhushan, Shashi; Ragunathan, Priya; Shin, Joon; Dick, Thomas; Grüber, Gerhard |