Browsing by Author Harikishore, Amaravadhi

Showing results 1 to 18 of 18
Issue DateTitleAuthor(s)
 2021Antiviral activity against Middle East Respiratory Syndrome coronavirus by Montelukast, an anti-asthma drugGan, Hanjie Jonathan; Harikishore, Amaravadhi; Lee, Jihye; Jeon, Sangeun; Rajan, Sreekanth; Chen, Ming Wei; Neo, Jun Long; Kim, Seungtaek; Yoon, Ho Sup
2022Atomic solution structure of Mycobacterium abscessus F-ATP synthase subunit ε and identification of Ep1MabF1 as a targeted inhibitorShin, Joon; Harikishore, Amaravadhi; Wong, Chui Fann; Ragunathan, Priya; Dick, Thomas; Grüber, Gerhard
2015Combination of pharmacophore hypothesis and molecular docking to identify novel inhibitors of HCV NS5B polymeraseHarikishore, Amaravadhi; Li, Enlin; Lee, Jia Jun; Cho, Nam-Joon; Yoon, Ho Sup
 2009Crystallographic structure of the tetratricopeptide repeat domain of Plasmodium falciparum FKBP35 and its molecular interaction with Hsp90 C-terminal pentapeptideAlag, Reema; Bharatham, Nagakumar; Dong, Aiping; Hills, Tanya; Harikishore, Amaravadhi; Widjaja, Anissa Anindya; Shochat, Susana Geifman; Hui, Raymond; Yoon, Ho Sup
2021Deciphering the role of ion channels in early defense signaling against herbivorous insectsGandhi, Akanksha; Kariyat, Rupesh; Harikishore, Amaravadhi; Ayati, Marzieh; Bhunia, Anirban; Sahoo, Nirakar
2020Discovery of a novel mycobacterial F-ATP synthase inhibitor and its potency in combination with diarylquinolinesHotra, Adam; Ragunathan, Priya; Ng, Pearly Shuyi; Seankongsuk, Pattarakiat; Harikishore, Amaravadhi; Sarathy, Jickky Palmae; Saw, Wuan-Geok; Lakshmanan, Umayal; Sae-Lao, Patcharaporn; Kalia, Nitin Pal; Shin, Joon; Kalyanasundaram, Revathy; Anbarasu, Sivaraj; Parthasarathy, Krupakar; Pradeep, Chaudhari Namrata; Makhija, Harshyaa; Dröge, Peter; Poulsen, Anders; Tan, Jocelyn Hui Ling; Pethe, Kevin; Dick, Thomas; Bates, Roderick Wayland; Grüber, Gerhard
2019Disrupting coupling within mycobacterial F-ATP synthases subunit ε causes dysregulated energy production and cell wall biosynthesisSaw, Wuan-Geok; Wu, Mu-Lu; Ragunathan, Priya; Biuković, Goran; Lau, Aik-Meng; Shin, Joon; Harikishore, Amaravadhi; Cheung, Chen-Yi; Hards, Kiel; Sarathy, Jickky Palmae; Bates, Roderick Wayland; Cook, Gregory M.; Dick, Thomas; Grüber, Gerhard
 2013The flavonoid myricetin reduces nocturnal melatonin levels in the blood through the inhibition of serotonin N-acetyltransferaseShin, Jae-Cheon; Jung, Hoe-Yune; Harikishore, Amaravadhi; Kwon, Oh-Deog; Yoon, Ho Sup; Kim, Kyong-Tai; Choi, Bo-Hwa
2014Luteolin suppresses cancer cell proliferation by targeting vaccinia-related kinase 1Kim, Ye Seul; Kim, Seong-Hoon; Shin, Joon; Harikishore, Amaravadhi; Lim, Jong-Kwan; Jung, Youngseob; Lyu, Ha-Na; Baek, Nam-In; Choi, Kwan Yong; Yoon, Ho Sup; Kim, Kyong-Tai
2022Mutational analysis of mycobacterial F‑ATP synthase subunit δ leads to a potent δ enzyme inhibitorHarikishore, Amaravadhi; Saw, Wuan-Geok; Ragunathan, Priya; Litty, Dennnis; Dick, Thomas; Müller, Volker; Grüber, Gerhard
 2012Solution structure of FK506-binding protein 12 from Aedes aegyptiChakraborty, Goutam; Shin, Joon; Nguyen, Quoc Toan; Harikishore, Amaravadhi; Baek, Kwanghee; Yoon, Ho Sup
2022Structural and mechanistic insights into Mycobacterium abscessus as-partate decarboxylase PanD and a pyrazinoic acid-derived inhibitorSaw, Wuan Geok; Leow, Chen Yen; Harikishore, Amaravadhi; Shin, Joon; Cole, Malcolm S.; Aragaw, Wassihun Wedajo; Ragunathan, Priya; Hegde, Pooja; Aldrich, Courtney C.; Dick, Thomas; Grüber, Gerhard
 2022Structure activity relationship of pyrazinoic acid analogs as potential antimycobacterial agentsHegde, Pooja V.; Aragaw, Wassihun W.; Cole, Malcolm S.; Jachak, Gorakhnath; Ragunathan, Priya; Sharma, Sachin; Harikishore, Amaravadhi; Grüber, Gerhard; Dick, Thomas; Aldrich, Courtney C.
2014Suprafenacine, an indazole-hydrazide agent, targets cancer cells through microtubule destabilizationChoi, Bo-Hwa; Chattopadhaya, Souvik; Feng, Lin; Nguyen, Quoc Toan; Lim, Chuan Bian; Harikishore, Amaravadhi; Nanga, Ravi Prakash Reddy; Bharatham, Nagakumar; Zhao, Yan; Yoon, Ho Sup; Thanh, Le Nguyen; Liu, Xuewei
2021A systematic assessment of mycobacterial F1-ATPase subunit ϵ’s role in latent ATPase hydrolysisWong, Chui-Fann; Lau, Aik-Meng; Harikishore, Amaravadhi; Saw, Wuan-Geok; Shin, Joon; Ragunathan, Priya; Bhushan, Shashi; Ngan, So-Fong Cam; Sze, Siu Kwan; Bates, Roderick Wayland; Dick, Thomas; Grüber, Gerhard
2021Targeting mycobacterial F-ATP synthase C-terminal α subunit interaction motif on rotary subunit γHarikishore, Amaravadhi; Wong, Chui-Fann; Ragunathan, Priya; Litty, Dennis; Müller, Volker; Grüber, Gerhard
2020Targeting the menaquinol binding loop of mycobacterial cytochrome bd oxidaseHarikishore, Amaravadhi; Chong, Sherilyn Shi Min; Ragunathan, Priya; Bates, Roderick Wayland; Grüber, Gerhard
2015Ursolic acid exerts anti-cancer activity by suppressing vaccinia-related kinase 1-mediated damage repair in lung cancer cellsKim, Seong-Hoon; Ryu, Hye Guk; Lee, Juhyun; Shin, Joon; Harikishore, Amaravadhi; Jung, Hoe-Youn; Kim, Ye Seul; Lyu, Ha-Na; Oh, Eunji; Baek, Nam-In; Choi, Kwan-Yong; Yoon, Ho Sup; Kim, Kyong-Tai